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Peptide History intermediate

History of Peptide Formulation Science

The development of formulation strategies for peptide stability and delivery.

By Encyclopeptide Editorial | 1 min read
formulation stability delivery history

Overview

Peptide formulation science has evolved to address the unique stability and delivery challenges of peptide therapeutics.

Key Developments

  • 1920s: Simple aqueous insulin formulations
  • 1950s: Protamine zinc insulin for extended action
  • 1970s: Lyophilized peptide formulations
  • 1980s: Depot injectable formulations
  • 1990s: PEGylation for half-life extension
  • 2000s: Nanoparticle and liposomal formulations
  • 2010s: Oral permeation enhancer technology

Impact

Formulation innovation has been as important as molecular design in enabling successful peptide therapeutics.

References

  • Source: ENCP Peptide Database
  • Category: Peptide History

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