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Peptide History beginner

History of Peptide-GLP-1 Development

The journey from GLP-1 discovery to blockbuster diabetes and obesity drugs.

By Encyclopeptide Editorial | 1 min read
glp-1 incretin diabetes obesity

Overview

GLP-1 receptor agonists have become the most commercially successful peptide drug class, transforming diabetes and obesity treatment.

Key Milestones

  • 1983: GLP-1 sequenced
  • 1990s: Incretin hypothesis established
  • 2002: Exendin-4 approved as exenatide
  • 2010: Liraglutide approved
  • 2017: Semaglutide approved
  • 2019: Oral semaglutide breakthrough
  • 2021: Semaglutide for obesity
  • 2023: Tirzepatide dual agonist

Impact

GLP-1 agonists represent a paradigm shift in metabolic medicine, with potential benefits extending to cardiovascular, liver, and kidney diseases.

References

  • Source: ENCP Peptide Database
  • Category: Peptide History

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