Skip to content
Peptide Modifications advanced

Peptide Prenylation Sites

Overview of farnesyl and geranylgeranyl modifications anchoring peptides to membranes.

By Encyclopeptide Editorial | 1 min read
prenylation lipid membrane modification

Overview

Prenylation attaches farnesyl (C15) or geranylgeranyl (C20) isoprenoid groups to C-terminal cysteine residues.

Types

  • Farnesylation: CAAX motif recognition by farnesyltransferase
  • Geranylgeranylation: Rab GGTase and GGTase-I modifications

Biological Significance

Prenylation is essential for Ras, Rho, and Rab GTPase membrane localization and function. Farnesyltransferase inhibitors were developed as anticancer agents.

References

  • Source: ENCP Peptide Database
  • Category: Peptide Modifications

Test Your Knowledge

Reinforce what you learned about Peptide Prenylation Sites with interactive quizzes on Wikipept.

Take a Quiz on Wikipept