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Pancreatic Peptides beginner

C-Peptide: Oligopeptide Research Reference

31-amino acid connecting peptide cleaved from proinsulin, used as a marker of endogenous insulin secretion. This peptide or oligopeptide is studied for its b...

By Encyclopeptide Editorial | 2 min read
proinsulin diabetes biomarker beta-cell-function

Chemical Identity

PropertyValue
Chemical FormulaC129H211N35O48
Molecular Weight3020 Da
CAS Number59401-28-4
Peptide ClassConnecting Peptide (31 amino acids)
SequenceEAEDLQVGQVELGGGPGAGSLQPLALEGSLQ

Structure

C-peptide is a 31-amino acid peptide that connects the A and B chains of proinsulin in the precursor molecule. During insulin biosynthesis, proinsulin is cleaved by prohormone convertases PC1/3 and PC2, releasing C-peptide and mature insulin in equimolar amounts.

Mechanism of Action

C-peptide was long considered biologically inactive, but evidence suggests it binds to a G-protein-coupled receptor (possibly CXCR4) on cell surfaces, activating eNOS and Na+/K+-ATPase. It may have beneficial effects on microvascular blood flow, nerve function, and renal function in type 1 diabetes.

Clinical Applications

  • Beta-cell function assessment: C-peptide levels reflect endogenous insulin production
  • Type 1 vs type 2 diabetes: Distinguishes insulin deficiency from resistance
  • Hypoglycemia evaluation: Factitious vs insulinoma
  • Research: Potential therapeutic in type 1 diabetes

Pharmacology

  • Half-life: 20-30 minutes (vs 3-5 min for insulin)
  • Molar ratio: 1:1 with insulin
  • Renal clearance: 5% of insulin clearance
  • Stability: More stable than insulin in blood samples

References

  • Steiner, D.F., & Oyer, P.E. (1967). The biosynthesis of insulin. Proceedings of the National Academy Sciences, 57, 473-480.
  • Wahren, J., et al. (2012). Role of C-peptide in human physiology. American Journal of Physiology, 298, E731-E740.

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